{"id":70508,"date":"2026-04-27T11:19:36","date_gmt":"2026-04-27T03:19:36","guid":{"rendered":"http:\/\/111.62.156.167\/?chemical-product=eltrombopag-acyl-glucuronide"},"modified":"2026-04-27T11:19:36","modified_gmt":"2026-04-27T03:19:36","slug":"eltrombopag-acyl-glucuronide","status":"publish","type":"chemical-product","link":"https:\/\/bio-get.com\/?chemical-product=eltrombopag-acyl-glucuronide","title":{"rendered":"Eltrombopag Acyl Glucuronide"},"content":{"rendered":"<p>\u4ea7\u54c1\u8bf4\u660e<br \/>\n\u4ea7\u54c1\u8bf4\u660e<br \/>\n1. \u4ea7\u54c1\u6982\u8ff0\u4e0e\u5316\u5b66\u7279\u6027<br \/>\nEltrombopag Acyl Glucuronide\uff08\u4ea7\u54c1\u76ee\u5f55\u53f7\uff1aBGGCB-4625\uff0cCAS\u53f7\uff1a1396009-05-4\uff09\u662f\u4e00\u79cd\u9170\u57fa\u8461\u8404\u7cd6\u919b\u9178\u4ee3\u8c22\u7269\uff0c\u5176\u5316\u5b66\u540d\u79f0\u4e3aEltrombopag\u7684\u8461\u8404\u7cd6\u919b\u9178\u7ed3\u5408\u7269\u3002\u8be5\u5316\u5408\u7269\u7684\u5206\u5b50\u5f0f\u4e3aC31H30N4O10\uff0c\u5206\u5b50\u91cf\u4e3a618.59 g\/mol\uff0c\u7eaf\u5ea6\u9ad8\u4e8e96%\u3002\u4f5c\u4e3a\u4e00\u79cd\u91cd\u8981\u7684\u4ee3\u8c22\u4ea7\u7269\uff0c\u5176\u7ed3\u6784\u7279\u5f81\u4e3aEltrombopag\u4e0e\u8461\u8404\u7cd6\u919b\u9178\u901a\u8fc7\u9170\u57fa\u952e\u7ed3\u5408\uff0c\u5177\u6709\u8f83\u9ad8\u7684\u6781\u6027\u548c\u6c34\u6eb6\u6027\uff0c\u9002\u7528\u4e8e\u4ee3\u8c22\u7814\u7a76\u548c\u836f\u7269\u5f00\u53d1\u9886\u57df\u3002<br \/>\n2. \u751f\u7269\u5316\u5b66\u529f\u80fd\u4e0e\u91cd\u8981\u6027<br \/>\nEltrombopag Acyl Glucuronide\u662fEltrombopag\uff08\u4e00\u79cd\u8840\u5c0f\u677f\u751f\u6210\u7d20\u53d7\u4f53\u6fc0\u52a8\u5242\uff09\u5728\u4f53\u5185\u7684\u4e3b\u8981\u4ee3\u8c22\u4ea7\u7269\u4e4b\u4e00\u3002\u5176\u5f62\u6210\u4f9d\u8d56\u4e8e\u809d\u810f\u4e2d\u7684UDP-\u8461\u8404\u7cd6\u919b\u9178\u8f6c\u79fb\u9176\uff08UGT\uff09\u4ecb\u5bfc\u7684\u8461\u8404\u7cd6\u919b\u9178\u5316\u53cd\u5e94\u3002\u8be5\u4ee3\u8c22\u4ea7\u7269\u5728\u836f\u7269\u4ee3\u8c22\u52a8\u529b\u5b66\u7814\u7a76\u4e2d\u5177\u6709\u91cd\u8981\u610f\u4e49\uff0c\u53ef\u7528\u4e8e\u8bc4\u4f30Eltrombopag\u7684\u4ee3\u8c22\u9014\u5f84\u3001\u751f\u7269\u8f6c\u5316\u6548\u7387\u4ee5\u53ca\u6f5c\u5728\u7684\u836f\u7269\u76f8\u4e92\u4f5c\u7528\u3002<br \/>\n3. \u4e3b\u8981\u5e94\u7528\u9886\u57df\u4e0e\u5177\u4f53\u7528\u9014<br \/>\n\u8be5\u5316\u5408\u7269\u5e7f\u6cdb\u5e94\u7528\u4e8e\u836f\u7406\u5b66\u548c\u6bd2\u7406\u5b66\u7814\u7a76\uff0c\u7279\u522b\u662f\u5728\u836f\u7269\u4ee3\u8c22\u4e0e\u6392\u6cc4\uff08ADME\uff09\u7814\u7a76\u4e2d\u4f5c\u4e3a\u6807\u51c6\u54c1\u6216\u5bf9\u7167\u54c1\u4f7f\u7528\u3002\u5177\u4f53\u7528\u9014\u5305\u62ec\uff1a<br \/>\n&#8211; 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