{"id":68489,"date":"2026-04-27T10:56:00","date_gmt":"2026-04-27T02:56:00","guid":{"rendered":"http:\/\/111.62.156.167\/?chemical-product=nilotinib"},"modified":"2026-04-27T10:56:00","modified_gmt":"2026-04-27T02:56:00","slug":"nilotinib","status":"publish","type":"chemical-product","link":"https:\/\/bio-get.com\/?chemical-product=nilotinib","title":{"rendered":"nilotinib"},"content":{"rendered":"<p>\u4ea7\u54c1\u8bf4\u660e<br \/>\n\u4ea7\u54c1\u8bf4\u660e<br \/>\n1. \u4ea7\u54c1\u6982\u8ff0\u4e0e\u5316\u5b66\u7279\u6027<br \/>\n\u5c3c\u6d1b\u66ff\u5c3c\uff08Nilotinib\uff09\u662f\u4e00\u79cd\u5c0f\u5206\u5b50\u916a\u6c28\u9178\u6fc0\u9176\u6291\u5236\u5242\uff0c\u5316\u5b66\u540d\u79f0\u4e3a4-\u7532\u57fa-N-[3-(4-\u7532\u57fa-1H-\u54aa\u5511-1-\u57fa)-5-(\u4e09\u6c1f\u7532\u57fa)\u82ef\u57fa]-3-[(4-\u5421\u5576-3-\u57fa\u5627\u5576-2-\u57fa)\u6c28\u57fa]\u82ef\u7532\u9170\u80fa\uff0cCAS\u53f7\u4e3a641571-10-0\u3002\u5176\u5206\u5b50\u5f0f\u4e3aC28H22F3N7O\uff0c\u5206\u5b50\u91cf\u4e3a529.516\uff0c\u7eaf\u5ea6\u9ad8\u4e8e96%\u3002\u8be5\u5316\u5408\u7269\u4e3a\u767d\u8272\u81f3\u7c7b\u767d\u8272\u7ed3\u6676\u6027\u7c89\u672b\uff0c\u53ef\u6eb6\u4e8e\u6709\u673a\u6eb6\u5242\u5982DMSO\uff0c\u5fae\u6eb6\u4e8e\u6c34\u3002<br \/>\n2. \u751f\u7269\u5316\u5b66\u529f\u80fd\u4e0e\u91cd\u8981\u6027<br \/>\n\u5c3c\u6d1b\u66ff\u5c3c\u662f\u4e00\u79cd\u9ad8\u6548\u7684Bcr-Abl\u916a\u6c28\u9178\u6fc0\u9176\u9009\u62e9\u6027\u6291\u5236\u5242\uff0c\u901a\u8fc7\u7ade\u4e89\u6027\u7ed3\u5408ATP\u7ed3\u5408\u4f4d\u70b9\uff0c\u963b\u65adBcr-Abl\u86cb\u767d\u7684\u5f02\u5e38\u6fc0\u6d3b\u3002\u5176\u6291\u5236\u4f5c\u7528\u5f3a\u4e8e\u4f0a\u9a6c\u66ff\u5c3c\uff0c\u5c24\u5176\u5bf9\u90e8\u5206\u4f0a\u9a6c\u66ff\u5c3c\u8010\u836f\u7a81\u53d8\u6709\u6548\u3002\u5c3c\u6d1b\u66ff\u5c3c\u5728\u7ec6\u80de\u4fe1\u53f7\u4f20\u5bfc\u8c03\u63a7\u4e2d\u53d1\u6325\u5173\u952e\u4f5c\u7528\uff0c\u80fd\u591f\u6291\u5236\u767d\u8840\u75c5\u7ec6\u80de\u7684\u589e\u6b96\u5e76\u8bf1\u5bfc\u5176\u51cb\u4ea1\u3002<br \/>\n3. \u4e3b\u8981\u5e94\u7528\u9886\u57df\u4e0e\u5177\u4f53\u7528\u9014<br \/>\n\u5c3c\u6d1b\u66ff\u5c3c\u4e3b\u8981\u7528\u4e8e\u6162\u6027\u9ad3\u6027\u767d\u8840\u75c5\uff08CML\uff09\u7684\u6cbb\u7597\uff0c\u5c24\u5176\u662f\u8d39\u57ce\u67d3\u8272\u4f53\u9633\u6027\uff08Ph+\uff09\u7684\u6162\u6027\u671f\u6216\u52a0\u901f\u671f\u60a3\u8005\u3002\u6b64\u5916\uff0c\u5b83\u4e5f\u7528\u4e8e\u79d1\u5b66\u7814\u7a76\u4e2d\uff0c\u4f5c\u4e3a\u7814\u7a76Bcr-Abl\u4fe1\u53f7\u901a\u8def\u53ca\u8010\u836f\u673a\u5236\u7684\u5206\u5b50\u5de5\u5177\u3002\u5728\u4f53\u5916\u5b9e\u9a8c\u4e2d\uff0c\u5c3c\u6d1b\u66ff\u5c3c\u53ef\u7528\u4e8e\u7ec6\u80de\u57f9\u517b\u6a21\u578b\uff0c\u4ee5\u8bc4\u4f30\u5176\u5bf9\u80bf\u7624\u7ec6\u80de\u751f\u957f\u7684\u5f71\u54cd\u3002<br \/>\n4. \u50a8\u5b58\u6761\u4ef6\u4e0e\u4f7f\u7528\u5efa\u8bae<br \/>\n\u5c3c\u6d1b\u66ff\u5c3c\u5e94\u5bc6\u5c01\u4fdd\u5b58\u4e8e-20\u00b0C\u5e72\u71e5\u73af\u5883\u4e2d\uff0c\u907f\u514d\u5149\u7167\u548c\u6f6e\u6e7f\u3002\u4f7f\u7528\u65f6\u9700\u5728\u65e0\u83cc\u6761\u4ef6\u4e0b\u64cd\u4f5c\uff0c\u5efa\u8bae\u6eb6\u89e3\u4e8eDMSO\u914d\u5236\u6210\u6bcd\u6db2\u540e\u8fdb\u4e00\u6b65\u7a00\u91ca\u3002\u5b9e\u9a8c\u8fc7\u7a0b\u4e2d\u9700\u4f69\u6234\u9632\u62a4\u624b\u5957\u548c\u53e3\u7f69\uff0c\u907f\u514d\u76f4\u63a5\u63a5\u89e6\u76ae\u80a4\u6216\u5438\u5165\u7c89\u5c18\u3002<br \/>\n5. \u8d28\u91cf\u63a7\u5236\u4e0e\u5b89\u5168\u4fe1\u606f<br \/>\n\u672c\u4ea7\u54c1\u7ecfHPLC\u68c0\u6d4b\uff0c\u7eaf\u5ea6>96%\uff0c\u7b26\u5408\u79d1\u7814\u7ea7\u6807\u51c6\u3002\u5c3c\u6d1b\u66ff\u5c3c\u5bf9\u4eba\u4f53\u6709\u5bb3\uff0c\u53ef\u80fd\u5bf9\u751f\u6b96\u7cfb\u7edf\u9020\u6210\u635f\u4f24\uff0c\u64cd\u4f5c\u65f6\u9700\u4e25\u683c\u9075\u5b88\u5b9e\u9a8c\u5ba4\u5b89\u5168\u89c4\u8303\u3002\u5e9f\u5f03\u7269\u5e94\u6309\u7167\u5371\u9669\u5316\u5b66\u54c1\u5904\u7406\u6d41\u7a0b\u5904\u7f6e\u3002\u5982\u9700\u8fdb\u4e00\u6b65\u6bd2\u7406\u5b66\u6570\u636e\uff0c\u8bf7\u53c2\u8003\u6750\u6599\u5b89\u5168\u6570\u636e\u8868\uff08MSDS\uff09\u3002<\/p>\n","protected":false},"featured_media":0,"template":"","meta":{"_acf_changed":false,"_kad_blocks_custom_css":"","_kad_blocks_head_custom_js":"","_kad_blocks_body_custom_js":"","_kad_blocks_footer_custom_js":"","_kadence_starter_templates_imported_post":false,"_kad_post_transparent":"","_kad_post_title":"","_kad_post_layout":"","_kad_post_sidebar_id":"","_kad_post_content_style":"","_kad_post_vertical_padding":"","_kad_post_feature":"","_kad_post_feature_position":"","_kad_post_header":false,"_kad_post_footer":false,"_kad_post_classname":""},"product_category":[31],"class_list":["post-68489","chemical-product","type-chemical-product","status-publish","hentry","product_category-31"],"acf":[],"taxonomy_info":{"product_category":[{"value":31,"label":"\u7cd6\u79d1\u5b66"}]},"featured_image_src_large":false,"author_info":[],"comment_info":"","_links":{"self":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/chemical-product\/68489","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/chemical-product"}],"about":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/types\/chemical-product"}],"wp:attachment":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=68489"}],"wp:term":[{"taxonomy":"product_category","embeddable":true,"href":"https:\/\/bio-get.com\/index.php?rest_route=%2Fwp%2Fv2%2Fproduct_category&post=68489"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}