{"id":68356,"date":"2026-04-27T10:54:30","date_gmt":"2026-04-27T02:54:30","guid":{"rendered":"http:\/\/111.62.156.167\/?chemical-product=palbociclib-isethionate"},"modified":"2026-04-27T10:54:30","modified_gmt":"2026-04-27T02:54:30","slug":"palbociclib-isethionate","status":"publish","type":"chemical-product","link":"https:\/\/bio-get.com\/?chemical-product=palbociclib-isethionate","title":{"rendered":"Palbociclib isethionate"},"content":{"rendered":"<p>\u4ea7\u54c1\u8bf4\u660e<br \/>\n### \u4ea7\u54c1\u8bf4\u660e<br \/>\n#### 1. \u4ea7\u54c1\u6982\u8ff0\u4e0e\u5316\u5b66\u7279\u6027<br \/>\nPalbociclib isethionate\uff08\u5316\u5b66\u540d\u79f0\uff1a\u5e15\u535a\u897f\u5c3c\u5f02\u786b\u4ee3\u786b\u9178\u76d0\uff09\u662f\u4e00\u79cd\u5c0f\u5206\u5b50\u6291\u5236\u5242\uff0c\u5316\u5b66\u5f0f\u4e3aC26H35N7O6S\uff0c\u5206\u5b50\u91cf\u4e3a573.664\uff0cCAS\u53f7\u4e3a827022-33-3\u3002\u672c\u54c1\u4e3a\u9ad8\u7eaf\u5ea6\u5316\u5408\u7269\uff0c\u7eaf\u5ea6>96%\uff0c\u5448\u767d\u8272\u81f3\u7c7b\u767d\u8272\u7c89\u672b\uff0c\u53ef\u6eb6\u4e8eDMSO\u7b49\u6709\u673a\u6eb6\u5242\uff0c\u5fae\u6eb6\u4e8e\u6c34\u3002\u5176\u7ed3\u6784\u4e2d\u7684\u5f02\u786b\u4ee3\u786b\u9178\u76d0\u5f62\u5f0f\u589e\u5f3a\u4e86\u6eb6\u89e3\u6027\u548c\u7a33\u5b9a\u6027\uff0c\u9002\u7528\u4e8e\u79d1\u7814\u548c\u836f\u7269\u5f00\u53d1\u9886\u57df\u7684\u5e94\u7528\u3002<br \/>\n#### 2. \u751f\u7269\u5316\u5b66\u529f\u80fd\u4e0e\u91cd\u8981\u6027<br \/>\nPalbociclib\u662f\u4e00\u79cd\u9009\u62e9\u6027CDK4\/6\uff08\u7ec6\u80de\u5468\u671f\u4f9d\u8d56\u6027\u6fc0\u91764\/6\uff09\u6291\u5236\u5242\uff0c\u901a\u8fc7\u963b\u65adRb\u86cb\u767d\u7684\u78f7\u9178\u5316\uff0c\u6291\u5236\u7ec6\u80de\u5468\u671f\u4eceG1\u671f\u5411S\u671f\u8fc7\u6e21\uff0c\u4ece\u800c\u6291\u5236\u80bf\u7624\u7ec6\u80de\u589e\u6b96\u3002\u8be5\u673a\u5236\u5728\u4e73\u817a\u764c\u7b49\u591a\u79cd\u764c\u75c7\u7684\u6cbb\u7597\u4e2d\u5177\u6709\u91cd\u8981\u4ef7\u503c\uff0c\u5c24\u5176\u662f\u4e0e\u6fc0\u7d20\u7597\u6cd5\u8054\u7528\u65f6\u6548\u679c\u663e\u8457\u3002\u5176\u5f02\u786b\u4ee3\u786b\u9178\u76d0\u5f62\u5f0f\u8fdb\u4e00\u6b65\u4f18\u5316\u4e86\u836f\u7269\u7684\u751f\u7269\u5229\u7528\u5ea6\u548c\u5236\u5242\u7a33\u5b9a\u6027\u3002<br \/>\n#### 3. \u4e3b\u8981\u5e94\u7528\u9886\u57df\u4e0e\u5177\u4f53\u7528\u9014<br \/>\n\u672c\u54c1\u4e3b\u8981\u7528\u4e8e\u80bf\u7624\u5b66\u7814\u7a76\uff0c\u7279\u522b\u662f\u4e73\u817a\u764c\u3001\u80ba\u764c\u548c\u5176\u4ed6\u5b9e\u4f53\u7624\u7684\u4f53\u5916\u548c\u4f53\u5185\u5b9e\u9a8c\u3002\u5177\u4f53\u7528\u9014\u5305\u62ec\uff1a<br \/>\n1. \u4f5c\u4e3aCDK4\/6\u6291\u5236\u5242\u7684\u9633\u6027\u5bf9\u7167\u5316\u5408\u7269\uff1b<br \/>\n2. \u7528\u4e8e\u7ec6\u80de\u5468\u671f\u8c03\u63a7\u673a\u5236\u7684\u7814\u7a76\uff1b<br \/>\n3. \u8054\u5408\u5176\u4ed6\u6297\u764c\u836f\u7269\uff08\u5982\u82b3\u9999\u9176\u6291\u5236\u5242\uff09\u8fdb\u884c\u534f\u540c\u6548\u5e94\u8bc4\u4f30\uff1b<br \/>\n4. \u836f\u7269\u4ee3\u8c22\u548c\u836f\u4ee3\u52a8\u529b\u5b66\uff08DMPK\uff09\u7814\u7a76\u3002<br \/>\n#### 4. \u50a8\u5b58\u6761\u4ef6\u4e0e\u4f7f\u7528\u5efa\u8bae<br \/>\n\u5efa\u8bae\u5c06\u672c\u54c1\u7f6e\u4e8e-20\u00b0C\u5e72\u71e5\u907f\u5149\u73af\u5883\u4e2d\u4fdd\u5b58\uff0c\u907f\u514d\u53cd\u590d\u51bb\u878d\u4ee5\u786e\u4fdd\u7a33\u5b9a\u6027\u3002\u4f7f\u7528\u65f6\u9700\u5728\u65e0\u83cc\u6761\u4ef6\u4e0b\u64cd\u4f5c\uff0c\u63a8\u8350\u4ee5DMSO\u914d\u5236\u6bcd\u6db2\uff08\u598210 mM\uff09\uff0c\u5e76\u5206\u88c5\u4fdd\u5b58\u4ee5\u51cf\u5c11\u964d\u89e3\u3002\u5de5\u4f5c\u6d53\u5ea6\u9700\u6839\u636e\u5b9e\u9a8c\u4f53\u7cfb\u4f18\u5316\uff0c\u901a\u5e38\u4f53\u5916\u5b9e\u9a8c\u6d53\u5ea6\u4e3a0.1-10 \u03bcM\u3002<br \/>\n#### 5. \u8d28\u91cf\u63a7\u5236\u4e0e\u5b89\u5168\u4fe1\u606f<br \/>\n\u672c\u54c1\u7ecfHPLC\u9a8c\u8bc1\u7eaf\u5ea6>96%\uff0c\u5e76\u63d0\u4f9bCOA\uff08\u8d28\u91cf\u5206\u6790\u8bc1\u4e66\uff09\u3002\u4f7f\u7528\u65f6\u9700\u9075\u5b88\u5b9e\u9a8c\u5ba4\u5b89\u5168\u89c4\u8303\uff0c\u907f\u514d\u76f4\u63a5\u63a5\u89e6\u76ae\u80a4\u6216\u5438\u5165\u7c89\u5c18\u3002\u64cd\u4f5c\u65f6\u4f69\u6234\u9632\u62a4\u624b\u5957\u3001\u53e3\u7f69\u53ca\u62a4\u76ee\u955c\u3002\u5982\u4e0d\u614e\u63a5\u89e6\uff0c\u7acb\u5373\u7528\u5927\u91cf\u6e05\u6c34\u51b2\u6d17\u5e76\u5c31\u533b\u3002\u5e9f\u5f03\u7269\u9700\u6309\u5371\u9669\u5316\u5b66\u54c1\u89c4\u5b9a\u5904\u7406\u3002<br \/>\n\u4ee5\u4e0a\u4fe1\u606f\u4ec5\u4f9b\u53c2\u8003\uff0c\u5177\u4f53\u5b9e\u9a8c\u65b9\u6848\u9700\u7ed3\u5408\u6587\u732e\u548c\u5b9e\u9645\u6761\u4ef6\u4f18\u5316\u3002<\/p>\n","protected":false},"featured_media":0,"template":"","meta":{"_acf_changed":false,"_kad_blocks_custom_css":"","_kad_blocks_head_custom_js":"","_kad_blocks_body_custom_js":"","_kad_blocks_footer_custom_js":"","_kadence_starter_templates_imported_post":false,"_kad_post_transparent":"","_kad_post_title":"","_kad_post_layout":"","_kad_post_sidebar_id":"","_kad_post_content_style":"","_kad_post_vertical_padding":"","_kad_post_feature":"","_kad_post_feature_position":"","_kad_post_header":false,"_kad_post_footer":false,"_kad_post_classname":""},"product_category":[31],"class_list":["post-68356","chemical-product","type-chemical-product","status-publish","hentry","product_category-31"],"acf":[],"taxonomy_info":{"product_category":[{"value":31,"label":"\u7cd6\u79d1\u5b66"}]},"featured_image_src_large":false,"author_info":[],"comment_info":"","_links":{"self":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/chemical-product\/68356","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/chemical-product"}],"about":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/types\/chemical-product"}],"wp:attachment":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=68356"}],"wp:term":[{"taxonomy":"product_category","embeddable":true,"href":"https:\/\/bio-get.com\/index.php?rest_route=%2Fwp%2Fv2%2Fproduct_category&post=68356"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}