{"id":22518,"date":"2026-04-01T18:41:55","date_gmt":"2026-04-01T10:41:55","guid":{"rendered":"http:\/\/111.62.156.167\/index.php\/product\/pacritinib\/"},"modified":"2026-04-01T22:26:20","modified_gmt":"2026-04-01T14:26:20","slug":"pacritinib","status":"publish","type":"chemical-product","link":"https:\/\/bio-get.com\/?chemical-product=pacritinib","title":{"rendered":"Pacritinib"},"content":{"rendered":"<p>\u4ea7\u54c1\u8bf4\u660e<br \/>\nPacritinib\u4ea7\u54c1\u8bf4\u660e\u4e66<br \/>\n1. \u4ea7\u54c1\u6982\u8ff0\u4e0e\u5316\u5b66\u7279\u6027<br \/>\nPacritinib\u662f\u4e00\u79cd\u5c0f\u5206\u5b50\u6fc0\u9176\u6291\u5236\u5242\uff0c\u5316\u5b66\u540d\u79f0\u4e3a(16E)-11-[2-(1-\u5421\u54af\u70f7\u57fa)\u4e59\u6c27\u57fa]-14,19-\u4e8c\u6c27\u6742-5,7,27-\u4e09\u6c2e\u6742\u56db\u73af[19.3.1.12,6.18,12]\u4e8c\u5341\u4e03\u78b3-1(25),2(27),3,5,8(26),9,11,16,21,23-\u5341\u70ef\u3002\u8be5\u5316\u5408\u7269\u5206\u5b50\u5f0f\u4e3aC28H32N4O3\uff0c\u5206\u5b50\u91cf472.579\uff0cCAS\u767b\u8bb0\u53f7\u4e3a937272-79-2\u3002\u672c\u54c1\u4e3a\u767d\u8272\u81f3\u7c7b\u767d\u8272\u7ed3\u6676\u7c89\u672b\uff0c\u7eaf\u5ea6\u7ecfHPLC\u6d4b\u5b9a\u5927\u4e8e96%\uff0c\u7b26\u5408\u751f\u5316\u8bd5\u5242\u6807\u51c6\u3002<br \/>\n2. \u751f\u7269\u5316\u5b66\u529f\u80fd\u4e0e\u91cd\u8981\u6027<br \/>\nPacritinib\u662f\u4e00\u79cd\u9009\u62e9\u6027JAK2\/FLT3\u53cc\u91cd\u6291\u5236\u5242\uff0c\u901a\u8fc7\u7279\u5f02\u6027\u9776\u5411JAK2\u7684JH1\u7ed3\u6784\u57df\u53d1\u6325\u4f5c\u7528\u3002\u5176\u72ec\u7279\u4e4b\u5904\u5728\u4e8e\u5bf9JAK2V617F\u7a81\u53d8\u4f53\u5177\u6709\u663e\u8457\u6291\u5236\u6d3b\u6027\uff0c\u540c\u65f6\u4fdd\u6301\u5bf9JAK1\u7684\u76f8\u5bf9\u9009\u62e9\u6027\uff0c\u8fd9\u4e00\u7279\u6027\u4f7f\u5176\u5728\u9aa8\u9ad3\u589e\u6b96\u6027\u80bf\u7624\u7814\u7a76\u4e2d\u5177\u6709\u91cd\u8981\u4ef7\u503c\u3002\u8be5\u5316\u5408\u7269\u8fd8\u80fd\u6709\u6548\u6291\u5236FLT3-ITD\u7a81\u53d8\uff0c\u663e\u793a\u51fa\u5e7f\u8c31\u6297\u80bf\u7624\u6f5c\u529b\u3002<br \/>\n3. \u4e3b\u8981\u5e94\u7528\u9886\u57df\u4e0e\u5177\u4f53\u7528\u9014<br \/>\n\u672c\u4ea7\u54c1\u4e3b\u8981\u5e94\u7528\u4e8e\u80bf\u7624\u5b66\u7814\u7a76\u9886\u57df\uff0c\u5177\u4f53\u5305\u62ec\uff1a\u4f5c\u4e3aJAK\/STAT\u4fe1\u53f7\u901a\u8def\u7814\u7a76\u7684\u5de5\u5177\u5316\u5408\u7269\uff1b\u7528\u4e8e\u9aa8\u9ad3\u7ea4\u7ef4\u5316\u3001\u6025\u6027\u9ad3\u7cfb\u767d\u8840\u75c5\u7b49\u8840\u6db2\u7cfb\u7edf\u6076\u6027\u80bf\u7624\u7684\u4f53\u5916\u7814\u7a76\uff1b\u5f00\u53d1\u65b0\u578b\u9776\u5411\u6cbb\u7597\u65b9\u6848\u7684\u4e34\u5e8a\u524d\u8bc4\u4f30\u3002\u5728\u836f\u7269\u7814\u53d1\u4e2d\uff0c\u5e38\u7528\u4e8e\u6fc0\u9176\u6291\u5236\u6d3b\u6027\u6d4b\u5b9a\u3001\u7ec6\u80de\u589e\u6b96\u6291\u5236\u5b9e\u9a8c\u548c\u52a8\u7269\u6a21\u578b\u7814\u7a76\u3002<br \/>\n4. \u50a8\u5b58\u6761\u4ef6\u4e0e\u4f7f\u7528\u5efa\u8bae<br \/>\n\u5efa\u8bae\u5c06\u672c\u54c1\u7f6e\u4e8e-20\u2103\u5e72\u71e5\u907f\u5149\u73af\u5883\u4e2d\u4fdd\u5b58\uff0c\u957f\u671f\u50a8\u5b58\u63a8\u8350\u4f7f\u7528\u60f0\u6027\u6c14\u4f53\u4fdd\u62a4\u3002\u4f7f\u7528\u65f6\u9700\u5728\u5e72\u71e5\u6c2e\u6c14\u73af\u5883\u4e0b\u64cd\u4f5c\uff0c\u6eb6\u89e3\u63a8\u8350\u4f7f\u7528DMSO\uff08\u6d53\u5ea6\u4e0d\u8d85\u8fc710mM\uff09\uff0c\u907f\u514d\u53cd\u590d\u51bb\u878d\u3002\u5de5\u4f5c\u6db2\u5e94\u5f53\u65e5\u914d\u5236\uff0c\u672a\u7528\u5b8c\u6eb6\u6db2\u5efa\u8bae\u4e22\u5f03\u3002\u672c\u54c1\u5bf9\u5149\u654f\u611f\uff0c\u5b9e\u9a8c\u8fc7\u7a0b\u5e94\u907f\u5149\u8fdb\u884c\u3002<br \/>\n5. \u8d28\u91cf\u63a7\u5236\u4e0e\u5b89\u5168\u4fe1\u606f<br \/>\n\u672c\u4ea7\u54c1\u7ecf\u4e25\u683c\u8d28\u63a7\uff0c\u5305\u62ecHPLC\u7eaf\u5ea6\u68c0\u6d4b\u3001\u8d28\u8c31\u9274\u5b9a\u548c\u6838\u78c1\u5171\u632f\u9a8c\u8bc1\u3002\u4f7f\u7528\u65f6\u9700\u4f69\u6234\u9632\u62a4\u88c5\u5907\uff0c\u907f\u514d\u5438\u5165\u6216\u76ae\u80a4\u63a5\u89e6\u3002MSDS\u6570\u636e\u663e\u793a\u8be5\u5316\u5408\u7269\u53ef\u80fd\u5177\u6709\u751f\u6b96\u6bd2\u6027\uff0c\u64cd\u4f5c\u5e94\u5728\u901a\u98ce\u6a71\u4e2d\u8fdb\u884c\u3002\u5e9f\u5f03\u7269\u5904\u7f6e\u9700\u7b26\u5408\u5371\u9669\u5316\u5b66\u54c1\u5904\u7406\u89c4\u8303\u3002\u4ec5\u4f9b\u79d1\u7814\u4f7f\u7528\uff0c\u4e0d\u9002\u7528\u4e8e\u4eba\u4f53\u6216\u517d\u533b\u4e34\u5e8a\u3002<\/p>\n","protected":false},"featured_media":7669,"template":"","meta":{"_acf_changed":false,"_kad_blocks_custom_css":"","_kad_blocks_head_custom_js":"","_kad_blocks_body_custom_js":"","_kad_blocks_footer_custom_js":"","_kadence_starter_templates_imported_post":false,"_kad_post_transparent":"","_kad_post_title":"","_kad_post_layout":"","_kad_post_sidebar_id":"","_kad_post_content_style":"","_kad_post_vertical_padding":"","_kad_post_feature":"","_kad_post_feature_position":"","_kad_post_header":false,"_kad_post_footer":false,"_kad_post_classname":""},"product_category":[17],"class_list":["post-22518","chemical-product","type-chemical-product","status-publish","has-post-thumbnail","hentry","product_category-17"],"acf":[],"taxonomy_info":{"product_category":[{"value":17,"label":"\u4e2d\u95f4\u4f53"}]},"featured_image_src_large":["https:\/\/bio-get.com\/wp-content\/uploads\/2026\/03\/937272-79-2.jpg",464,464,false],"author_info":[],"comment_info":"","_links":{"self":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/chemical-product\/22518","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/chemical-product"}],"about":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/types\/chemical-product"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/bio-get.com\/index.php?rest_route=\/wp\/v2\/media\/7669"}],"wp:attachment":[{"href":"https:\/\/bio-get.com\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=22518"}],"wp:term":[{"taxonomy":"product_category","embeddable":true,"href":"https:\/\/bio-get.com\/index.php?rest_route=%2Fwp%2Fv2%2Fproduct_category&post=22518"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}